ʻO Artesunate kahi lāʻau antimalarial maikaʻi e mālama ai i ka maʻi maʻi i hoʻokumu ʻia e Plasmodium falciparum. Pepehi ia i nā parasite no ka pale ʻana i ka maʻi a hoʻopau koke i nā hōʻailona pili i ka maʻi malaria, e like me ke kuni, ke poʻo, ke anuanu, ka ʻeha ʻiʻo, a me ka anemia. Hōʻike pū ʻo Artesunate i ka palekana kiʻekiʻe i nā noi lapaʻau.
Hana
ʻO Artesunate kahi lāʻau antimalarial maikaʻi loa e pepehi koke i nā parasites Plasmodium falciparum, me nā ʻano chloroquine-resistant strains. Hoʻohana ʻia ia e mālama i nā maʻi maʻi malaria, e hoʻēmi ana i nā hōʻailona e like me ke kuni, ke poʻo, a me ke anu, a me ke kōkua ʻana e pale i ka piʻi ʻana o ka maʻi. Ua hōʻike ʻia ʻo Artesunate i ka maikaʻi loa i nā hihia weliweli o ka maʻi malaria.
Palapala hōʻoia
Nā mea
Nā koi
Nā hualoaʻa
ʻO Dwehewehe
ʻAno:
ʻO ke aniani nila keʻokeʻo, ʻaʻala ʻole, ʻono ʻawaʻawa
Conforms
Ka hoʻoheheʻe
Fhiki ke hoʻoheheʻe ʻia i loko o ka chloroform; hiki ke hoʻoheheʻe ʻia i ka acetone, hiki ke hoʻoheheʻe ʻia i ka methanol a i ʻole ethanol; ʻaʻole hiki ke hoʻoheheʻe ʻia i ka wai
Kūlike
Lae hehee
145~150℃,mepalaho
146.3~146.8℃
ʻIkepili
Pane kala
Ahana ʻia ka waihoʻoluʻu ʻulaʻula
Conforms
Pane kala
Ahana ʻia ka waihoʻoluʻu ʻulaʻula e loli mālie a ʻeleʻele ke kū
Conforms
ʻO ka hoʻololi ʻana
Pono e hōʻike i nā waiwai optical dextral
Kūlike
A ME
Infrared absorption spectrum o ka ho'āʻo a me ka maʻamau(a i ʻoleinfrared reference spectra No. 220) he concordant
Kūlike
Hoao
1)Rmea ʻoluʻolu
(TLC)
SPono e loaʻa i kahi kikoʻī me ka hoʻonā (2).Kekahi wahi i loaa mekuhikuhihoʻonā, ʻokoʻa ka wahi nui,aole i oi aku mamua o ka hookahi, aisʻaʻole i ʻoi aku ka ikaika ma mua oka wahi nuiloaʻa me ka hoʻonā(1)(2.0%).
Conforms
2) Nalo ma ka maloʻo
≤ 0.5%
0.29%
3) KoenamaʻĀpana
≤ 0.1%
0.07%
4) Metala kaumaha(TLC)
≤ 10ppm
Conforms
ʻIke (ma ka driedkumu)
98.0%~102.0%(HPLC)
99.3%
Ka hopena:Kūlike ka huahana meCh.P.2010
Palapala noi
Hoʻohana mua ʻia ʻo Artesunate i ka mālama ʻana i nā maʻi maʻi malaria i hoʻokumu ʻia e ka Plasmodium falciparum parasite. ʻO kona ikaika e kūʻē i nā chloroquine-resistant strains e lilo ia i koho lapaʻau koʻikoʻi, ʻoi aku hoʻi i nā wahi i laha ʻia ai ka pale ʻana i ka maʻi malaria i nā lāʻau ʻē aʻe. Hāʻawi ʻia ʻo Artesunate i nā poʻe maʻi me ka maʻi maʻi e pepehi koke i nā parasites, hoʻomaha i nā hōʻailona e like me ke kuni, ke poʻo, ke anuanu, a me ka ʻeha ʻiʻo. I nā hihia koʻikoʻi o ka maʻi maʻi, hiki ke hoʻohana ʻia ka artesunate me ka intravenously e hoʻokō i nā hopena wikiwiki a ʻoi aku ka maikaʻi. Hoʻonui ʻia kāna mau noi i nā pākeke a me nā keiki, me ka hoʻoponopono ʻana i ka dosage kūpono e pili ana i ka makahiki a me ke kaumaha.